Bongarzone, Salvatore; Tran, Hoang Ngoc Ai; Cavalli, Andrea; Roberti, Marinella; Carloni, Paolo; Legname, Giuseppe; Bolognesi, Maria Laura
(American Chemical Society, 2010-11)
A library of 11 entries, featuring a 2,5-diamino-1,4-benzoquinones nucleus as spacer connecting two aromatic prion recognition motifs, was designed and evaluated against prion infection. Notably, 6-chloro-1,2,3,4-tetrahy ...